KDM5A-IN-1

Chemical Structure : KDM5A-IN-1

CAS No.: 1905481-36-8

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货号: PC-42028Not For Human Use, Lab Use Only.

KDM5A-IN-1 is a potent, orally bioavailable histone lysine demethylases 5 (KDM5) inhibitor with IC50 of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively.

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25 mg	￥5980	In stock
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生物&药学活性

KDM5A-IN-1 is a potent, orally bioavailable histone lysine demethylases 5 (KDM5) inhibitor with IC50 of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively.

KDM5A-IN-1 shows EC50 value of 960 nM for PC9 H3K4Me3, and less potent against other KDM enzymes (1A, 2B, 3B, 4C, 6A, 7B).

物理化学性质&存储条件

分子量	290.3608
分子式	C15H22N4O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Cyclopropanecarboxamide, N-[(3R)-1-[[5-(1-methylethyl)-1H-pyrazol-3-yl]carbonyl]-3-pyrrolidinyl]-

参考文献

1. Kwong Wah LAI, et al. WO 2016057924 A1 20160414.

KDM5A-IN-1

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物理化学性质&存储条件

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KDM5A-IN-1

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