KDM2A/7A inhibitor 1 |CAS:2169272-46-0 Probechem Biochemicals

Chemical Structure : KDM2A/7A inhibitor 1

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KDM2A/7A inhibitor 1 (KDM2A/7A-IN-1)

货号: PC-61815Not For Human Use, Lab Use Only.

KDM2A/7A inhibitor 1 is a potent, highly selective and cell-active inhibitor of KDM2A/7A with IC50 of 0.16 and 0.19 uM, respectively.

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生物&药学活性

KDM2A/7A inhibitor 1 is a potent, highly selective and cell-active inhibitor of KDM2A/7A with IC50 of 0.16 and 0.19 uM, respectively.
KDM2A/7A inhibitor 1 displays >75 fold selectivity towards KDM2A/7A versus other JmjC lysine demethylase.
KDM2A/7A inhibitor 1 shows cytotoxicity towards HeLa and HAP1 cells with EC50 of 22 uM and 7.1 uM respectively.

物理化学性质&存储条件

分子量	506.694
分子式	C33H38N4O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S,3S)-1-acetyl-3-phenyl-2-(5-(7-(pyrrolidin-1-yl)heptyl)pyridin-3-yl)indoline-3-carbonitrile

参考文献

1. Gerken P, et al. Angew Chem Int Ed Engl. 2017 Oct 4. doi: 10.1002/anie.201706788.

KDM2A/7A inhibitor 1 (KDM2A/7A-IN-1)

生物&药学活性

物理化学性质&存储条件

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KDM2A/7A inhibitor 1 (KDM2A/7A-IN-1)

生物&药学活性

物理化学性质&存储条件

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