JTE907 |CAS:282089-49-0 Probechem Biochemicals

Chemical Structure : JTE907

CAS No.: 282089-49-0

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JTE907 (JTE-907;JTE 907)

货号: PC-60763Not For Human Use, Lab Use Only.

JTE907 (JTE-907) is a potent, selective, orally active cannabinoid CB2 receptor inverse agonist with Ki of 35.9, 1.55 and 0.38 nM for human, mouse and rat CB2, respectively.

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5 mg	￥2180	In stock
10 mg	￥3580	In stock
25 mg	￥5680	In stock
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100 mg		Get quote

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生物&药学活性

JTE907 (JTE-907) is a potent, selective, orally active cannabinoid CB2 receptor inverse agonist with Ki of 35.9, 1.55 and 0.38 nM for human, mouse and rat CB2, respectively.
JTE907 increases of forskolin-stimulated cAMP production in CHO cells expressing CB2 in vitro, inhibits carrageenin-induced mouse paw edema dose dependently in mice.

物理化学性质&存储条件

分子量	438.48
分子式	C24H26N2O6
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(1,3-Benzodioxol-5-ylmethyl)-1,2-dihydro-7-methoxy-2-oxo-8-(pentyloxy)-3-quinolinecarboxamide

参考文献

1. Iwamura H, et al. J Pharmacol Exp Ther. 2001 Feb;296(2):420-5.

2. Ueda Y, et al. Eur J Pharmacol. 2005 Sep 27;520(1-3):164-71.

3. Maekawa T, et al. Eur J Pharmacol. 2006 Aug 7;542(1-3):179-83.

JTE907 (JTE-907;JTE 907)

生物&药学活性

物理化学性质&存储条件

参考文献

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JTE907 (JTE-907;JTE 907)

生物&药学活性

物理化学性质&存储条件

参考文献

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