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首页-小分子抑制剂&激动剂-GPCR-Ghrelin Receptor (GHSR)-JMV 2959
JMV 2959

Chemical Structure : JMV 2959

CAS No.: 925238-89-7

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JMV 2959 (JMV-2959, AEZS-123)

货号: PC-61828Not For Human Use, Lab Use Only.

JMV 2959 (AEZS-123) is a potent ghrelin receptor (GHS-R1A) antaognist with binding IC50 of 32 nM.

规格 价格 库存 数量
5 mg ￥1280 In stock
10 mg ￥1980 In stock
25 mg ￥3480 In stock
50 mg ￥5480 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

JMV 2959 (JMV-2959, AEZS-123) is a potent ghrelin receptor (GHS-R1A) antaognist with binding IC50 of 32 nM.
JMV 2959 suppresses ghrelin-induced and fasting-induced food intake at the level of the central nervous system.
JMV 2959 attenuates the NMDAR antagonist, phencyclidine-induced impairments in prepulse inhibition in rats.

物理化学性质&存储条件

分子量 508.626
分子式 C30H32N6O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-Amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]ethyl]acetamide

参考文献

1. Salomé N, et al. Eur J Pharmacol. 2009 Jun 10;612(1-3):167-73.

2. Landgren S, et al. Addict Biol. 2012 Jan;17(1):86-94.

3. Engel JA, et al. Psychopharmacology (Berl). 2015 Dec;232(23):4285-92.

4. Moulin A, et al. Amino Acids. 2013 Feb;44(2):301-14.

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