JKC-363 | MC4R antagonist | Probechem Biochemicals

Chemical Structure : JKC-363

CAS No.: 436083-30-6

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货号: PC-22664Not For Human Use, Lab Use Only.

JKC-363 (JKC363) is a highly potent, selective melanocortin MC4 receptor antagonist with IC50 of 0.5 nM, 90-fold selective over MC3 receptor.

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JKC-363 (JKC363) is a highly potent, selective melanocortin MC4 receptor antagonist with IC50 of 0.5 nM, 90-fold selective over MC3 receptor.

分子量	1506.71
分子式	C69H91N19O16S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(cyclic [Mpr11, D-Nal14, Cys18, Asp22-NH2]-beta-MSH11-22

1. Kim RY, et al. Biochem Biophys Res Commun. 2005 Apr 22;329(4):1178-85.

2. Doghman M, et al. Endocrinology. 2004 Feb;145(2):541-7.