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首页-小分子抑制剂&激动剂-GPCR-Ghrelin Receptor (GHSR)-Ibutamoren mesylate
Ibutamoren mesylate

Chemical Structure : Ibutamoren mesylate

CAS No.: 159752-10-0

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Ibutamoren mesylate (MK-677, MK-0677, L-163191)

货号: PC-45866Not For Human Use, Lab Use Only.

Ibutamoren mesylate (MK-0677) is a non-peptidic, poten and selective, orally-active agonist of the ghrelin receptor (GHSR) with EC50 of 1.3 nM (releases GH from rat pituitary cells).

规格 价格 库存 数量
10 mg ￥580 In stock
25 mg ￥980 In stock
50 mg ￥1580 In stock
100 mg ￥2280 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Ibutamoren mesylate (MK-0677) is a non-peptidic, poten and selective, orally-active agonist of the ghrelin receptor (GHSR) with EC50 of 1.3 nM (releases GH from rat pituitary cells).
Ibutamoren mesylate (MK-0677) significantly increased peak GH concentrations 20.4-fold at 0.25 mg/kg in beagles.
Ibutamoren mesylate (MK-0677) has shown to sustain activation of GH-IGF-1 Axis and increase in lean body mass but no change in total fat mass or visceral fat.

物理化学性质&存储条件

分子量 624.7692
分子式 C28H40N4O8S2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Propanamide, 2-amino-N-[(1R)-2-[1,2-dihydro-1-(methylsulfonyl)spiro[3H-indole-3,4'-piperidin]-1'-yl]-2-oxo-1-[(phenylmethoxy)methyl]ethyl]-2-methyl-, methanesulfonate (1:1)

参考文献

1. Patchett AA, et al. Proc Natl Acad Sci U S A. 1995 Jul 18;92(15):7001-5.

2. Jacks T, et al. Endocrinology. 1996 Dec;137(12):5284-9.

3. Copinschi G, et al. Neuroendocrinology. 1997 Oct;66(4):278-86.

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