HTS 01037 |CAS:682741-29-3 Probechem Biochemicals

Chemical Structure : HTS 01037

CAS No.: 682741-29-3

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HTS 01037 (HTS01037;HTS-01037)

货号: PC-61186Not For Human Use, Lab Use Only.

HTS01037 is a highly potent ligand of adipocyte fatty acid binding protein (A-FABP/aP2) with Ki of 0.67 uM.

规格	价格	库存
10 mg	￥1280	In stock
25 mg	￥1980	In stock
50 mg	￥3380	In stock
100 mg		Get quote

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生物&药学活性

HTS01037 is a highly potent ligand of adipocyte fatty acid binding protein (A-FABP/aP2) with Ki of 0.67 uM.
HTS 01037 competes with fatty acids for functional binding in the ligand-binding cavity of A-FABP/aP2, antagonizes the protein-protein interaction of A-FABP/aP2 with hormone sensitive lipase in cultured C8PA lipocytes at 10 uM.
HTS 01037 inhibits lipolysis in 3T3L1 adipocytes and reduces lipopolysaccharide-stimulated inflammation in bone marrow-derived macrophages.

物理化学性质&存储条件

分子量	337.364
分子式	C14H11NO5S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	[2,2'-Bithiophene]-5-carboxylic acid, 4-[(3-carboxy-1-oxo-2-propenyl)amino]-, 5-methyl ester (9CI)

参考文献

1. Hertzel AV, et al. J Med Chem. 2009 Oct 8;52(19):6024-31.

2. Steen KA, et al. Mol Cell Biol. 2017 Jan 4;37(2). pii: e00282-16.

3. Boss M, et al. Atherosclerosis. 2015 Jun;240(2):424-30.

HTS 01037 (HTS01037;HTS-01037)

生物&药学活性

物理化学性质&存储条件

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HTS 01037 (HTS01037;HTS-01037)

生物&药学活性

物理化学性质&存储条件

参考文献

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