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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-11β-HSD-HEAL-116
HEAL-116

Chemical Structure : HEAL-116

CAS No.: 3059767-85-7

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HEAL-116 (HEAL116)

货号: PC-24810Not For Human Use, Lab Use Only.

HEAL-116 is a potent, selective 3β-hydroxysteroid dehydrogenase type 1 (3βHSD1) inhibitor, shows binding specificity to the substrate-binding pocket of 3βHSD1 and effectively neutralizes the local charge environment.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

HEAL-116 is a potent, selective 3β-hydroxysteroid dehydrogenase type 1 (3βHSD1) inhibitor, shows binding specificity to the substrate-binding pocket of 3βHSD1 and effectively neutralizes the local charge environment.
HEAL-116 robustly inhibits 3βHSD1 activity and exerts pronounced antitumor effect in biochemical, cellular, and mouse models.

物理化学性质&存储条件

分子量 371.82
分子式 C20H18ClNO4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

3-(4-Chloro-3-(morpholinomethyl) phenyl)-7-hydroxy-4H-chromen-4-one

参考文献

1. He D, et al. Proc Natl Acad Sci U S A. 2025 Jul;122(26):e2422267122.

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