Guangxitoxin 1E | Kv2 channel inhibitor | Probechem Biochemicals

Chemical Structure : Guangxitoxin 1E

CAS No.: 1233152-82-3

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Guangxitoxin 1E (Guangxitoxin 1E TFA)

货号: PC-21704Not For Human Use, Lab Use Only.

Guangxitoxin 1E is a potent, specific inhibitor of Kv2.1 (KCNB1) and Kv2.2 with IC50 of 1-3 nM, has no significant effect on KV1.2, KV1.3, KV1.5, KV3.2 and BK potassium channels, also inactive against calcium and sodium channels CaV1.2, CaV2.2, NaV1.5, NaV1.7, NaV1.8.

规格	价格	库存
200 ug	￥2480	In stock
500 ug	￥3980	In stock
1 mg	￥5980	In stock
5 mg		Get quote

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生物&药学活性

Guangxitoxin 1E is a potent, specific inhibitor of Kv2.1 (KCNB1) and Kv2.2 with IC50 of 1-3 nM, has no significant effect on KV1.2, KV1.3, KV1.5, KV3.2 and BK potassium channels, also inactive against calcium and sodium channels CaV1.2, CaV2.2, NaV1.5, NaV1.7, NaV1.8.

物理化学性质&存储条件

分子量	3948.6
分子式	C178H248N44O45S7
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Glu-Gly-Glu-Cys-Gly-Gly-Phe-Trp-Trp-Lys-Cys-Gly-Ser-Gly-Lys-Pro-Ala-Cys-Cys-Pro-Lys-Tyr-Val-Cys-Ser-Pro-Lys-Trp-Gly-Leu-Cys-Asn-Phe-Pro-Met-Pro (Disulfide bridge:Cys4-Cys19;Cys11-Cys24;Cys18-Cys31)

参考文献

1. Herrington J, et al. Diabetes. 2006 Apr;55(4):1034-42.

Guangxitoxin 1E (Guangxitoxin 1E TFA)

生物&药学活性

物理化学性质&存储条件

参考文献

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Guangxitoxin 1E (Guangxitoxin 1E TFA)

生物&药学活性

物理化学性质&存储条件

参考文献

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