欢迎访问ProbeChem中文网站,英文网站请访问www.probechem.com

首页-小分子抑制剂&激动剂-Others-Other Targets-GlpG inhibitor 11
GlpG inhibitor 11

Chemical Structure : GlpG inhibitor 11

CAS No.:

GlpG inhibitor 11 (Rhomboid protease inhibitor)

货号: PC-60493Not For Human Use, Lab Use Only.

A potent, selective, reversible rhomboid proteases inhibitor with Ki of 45 nM for GlpG .

规格 价格 库存 数量

大包装,大折扣!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

A potent, selective, reversible rhomboid proteases inhibitor with Ki of 45 nM for GlpG ; does not inhibit most of the human serine hydrolases with the exception of PRCP and DPP7; potently inhibits endogenous GlpG in living E.coli. with IC50 of 2.7 nM.

物理化学性质&存储条件

分子量 855.015
分子式 C39H62N14O8
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(S)-2-(2-((S)-1-(((S)-3,4-dioxo-4-((4-phenylbutoxy)amino)butan-2-yl)amino)-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl)hydrazinyl)-5-guanidino-N-((S)-1-(((S)-1-guanidino-5,6-dioxoheptan-4-yl)amino)-3-methyl-1-oxobutan-2-yl)pentanamide

参考文献

1. Tichá A, et al. Cell Chem Biol. 2017 Dec 21;24(12):1523-1536.e4.

备案号:沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

联系我们 sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

询单

  • *产品名称:
  • *姓名:
  • *邮箱:
  • *公司名称:
  • *询单数量:
  • *国籍:
  • 询单信息: