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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Phospholipase-Giripladib
Giripladib

Chemical Structure : Giripladib

CAS No.: 865200-20-0

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Giripladib (PLA-695, PLA695)

货号: PC-22786Not For Human Use, Lab Use Only.

Giripladib (PLA-695) is a potent, specific cytoplasmic phospholipase A2 (cPLA2).
PLA-695 inhibits radiation induced phosphorylation of ERK and Akt in cultured endothelial cells.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Giripladib (PLA-695) is a potent, specific cytoplasmic phospholipase A2 (cPLA2).
PLA-695 inhibits radiation induced phosphorylation of ERK and Akt in cultured endothelial cells.
PLA-695 in combination with irradiation prevented endothelial cell migration.
PLA-695 enhanced radiation induced cell death and attenuated invasion of lung cancer cells.
PLA-695 inhibited the formation of new blood vessels and angiogenesis.

物理化学性质&存储条件

分子量 745.25
分子式 C41H36ClF3N2O4S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-(3-(1-benzhydryl-5-chloro-2-(2-(((2-(trifluoromethyl)phenyl)methyl)sulfonamido)ethyl)-1H-indol-3-yl)propyl)benzoic acid

参考文献

1. Thotala D, et al. PLoS One. 2013 Jul 19;8(7):e69688.

2. Duvernay MT, et al. Biochemistry. 2015 Sep 15;54(36):5578-88.

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