GYKI 52466 dihydrochloride |CAS:102771-26-6 Probechem Biochemicals

Chemical Structure : GYKI 52466 dihydrochloride

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GYKI 52466 dihydrochloride (GYKI52466 dihydrochloride)

货号: PC-61725Not For Human Use, Lab Use Only.

GYKI 52466 is a selective, non-competitive, orally active AMPA receptor (AMPAR) antagonist with IC50 of 10-20 uM against AMPA-induced responses.

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生物&药学活性

GYKI 52466 is a selective, non-competitive, orally active AMPA receptor (AMPAR) antagonist with IC50 of 10-20 uM against AMPA-induced responses.
GYKI 52466 displays >20-fold selectivity over kainate and NMDA receptors.
GYKI 52466 shows anticonvulsant and neuroprotective properties.

物理化学性质&存储条件

分子量	366.24
分子式	C17H15N3O2.2HCl
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(8-Methyl-9H-1,3-dioxolo[4,5-h][2,3]benzodiazepin-5-yl)-benzenamine dihydrochloride

参考文献

1. Tarnawa I, et al. Eur J Pharmacol. 1989 Aug 22;167(2):193-9.

2. Ouardouz M, et al. Neurosci Lett. 1991 Apr 15;125(1):5-8.

3. Donevan SD, et al. Neuron. 1993 Jan;10(1):51-9.

GYKI 52466 dihydrochloride (GYKI52466 dihydrochloride)

生物&药学活性

物理化学性质&存储条件

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GYKI 52466 dihydrochloride (GYKI52466 dihydrochloride)

生物&药学活性

物理化学性质&存储条件

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