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首页-小分子抑制剂&激动剂-GPCR-Free Fatty Acid Receptor (FFAR)-GW9508
GW9508

Chemical Structure : GW9508

CAS No.: 885101-89-3

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GW9508 (GW 9508)

货号: PC-20427Not For Human Use, Lab Use Only.

GW9508 (GW 9508) is a potent and selective FFA1 (GPR40) agonist with pEC50 of 7.32, >1,000-fold selectivity over FFA2 and FFA3 receptors.

规格 价格 库存 数量
25 mg ￥880 In stock
50 mg ￥1280 In stock
100 mg ￥2180 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GW9508 (GW 9508) is a potent and selective FFA1 (GPR40) agonist with pEC50 of 7.32, >1,000-fold selectivity over FFA2 and FFA3 receptors.
GW9508 dose dependently potentiated glucose-stimulated insulin secretion in MIN6 cells, but not in primary rat or mouse islets.
GW9508 potentiate the KCl-mediated increase in insulin secretion in MIN6 cells.
GW9508 suppresses CFA-induced inflammatory chronic pain in vivo.

物理化学性质&存储条件

分子量 347.41
分子式 C22H21NO3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-[[(3-Phenoxyphenyl)methyl]amino]benzenepropanoic acid

参考文献

1. Briscoe CP, et al. Br J Pharmacol. 2006 Jul;148(5):619-28.

2. Tikhonova IG, et al. J Med Chem. 2007 Jun 28;50(13):2981-9.

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