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首页-小分子抑制剂&激动剂-Cell Cycle/DNA Damage-Polo-like Kinase (PLK)-GW843682X
GW843682X

Chemical Structure : GW843682X

CAS No.: 660868-91-7

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GW843682X (GW 843682X;GW843682;GW-843682X)

货号: PC-42779Not For Human Use, Lab Use Only.

GW843682X is a potent and selective inhibitor of PLK1 (IC5=2.2 nM) and PLK3 (IC50=9 nM).

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10 mg ￥980 In stock
25 mg ￥1480 In stock
50 mg ￥2380 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GW843682X is a potent and selective inhibitor of PLK1 (IC5=2.2 nM) and PLK3 (IC50=9 nM).
GW843682X displays >1,000-fold lower than cell CDK-2/cyclin A, CDK1/cyclin A and aurora A.
GW843682X induces a transient G2-M arrest, mitotic spindle defects, and a multinucleate phenotype.

物理化学性质&存储条件

分子量 477.4562
分子式 C22H18F3N3O4S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-Thiophenecarboxamide, 5-(5,6-dimethoxy-1H-benzimidazol-1-yl)-3-[[2-(trifluoromethyl)phenyl]methoxy]-

参考文献

1. Lansing TJ, et al. Mol Cancer Ther. 2007 Feb;6(2):450-9.

2. Nihal M, et al. Cell Cycle. 2011 Apr 15;10(8):1303-11.

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