GSK962040 | Motilin receptor agonist | Probechem Biochemicals

Chemical Structure : GSK962040

CAS No.: 923565-21-3

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GSK962040 (Camicinal, GSK-962040)

货号: PC-42738Not For Human Use, Lab Use Only.

GSK962040 (Camicinal) is a potent, selective, small molecule motilin receptor agonist with pEC50 of 7.9 (hMTL-R).

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5 mg	￥2380	In stock
10 mg	￥3880	In stock
25 mg	￥5980	In stock
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

GSK962040 (Camicinal) is a potent, selective, small molecule motilin receptor (GPR38) agonist with pEC50 of 7.9 (hMTL-R).
GSK962040 displays selectivity over closely related human ghrelin acceptor (pEC50< 6.0) and no liabilities at the hERG channel.
GSK962040 possesses highly excellent pharmacokinetic profiles in both rat and dog.

物理化学性质&存储条件

分子量	424.5541
分子式	C25H33FN4O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: 12.73 mg/mL (Need ultrasonic)
Chemical Name/SMILES	Ethanone, 1-[4-[(3-fluorophenyl)amino]-1-piperidinyl]-2-[4-[[(3S)-3-methyl-1-piperazinyl]methyl]phenyl]-

参考文献

1. Westaway SM, et al. J Med Chem. 2009 Feb 26;52(4):1180-9.

2. Sanger GJ, et al. Neurogastroenterol Motil. 2009 Jun;21(6):657-64, e30-1.

3. Broad J, et al. Br J Pharmacol. 2012 Oct;167(4):763-74.

GSK962040 (Camicinal, GSK-962040)

生物&药学活性

物理化学性质&存储条件

参考文献

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GSK962040 (Camicinal, GSK-962040)

生物&药学活性

物理化学性质&存储条件

参考文献

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