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首页-小分子抑制剂&激动剂-Epigenetics-Bromodomain-GSK852
GSK852

Chemical Structure : GSK852

CAS No.: 2305842-30-0

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GSK852 (GSK-852)

货号: PC-72183Not For Human Use, Lab Use Only.

GSK852 (GSK-852) is a highly potent, second bromodomain (BD2)-selective BET inhibitor with pIC50 7.9 (BRD4 BD2), 1260-fold selectivity over BRD4 BD1.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    GSK852 (GSK-852) is a highly potent, second bromodomain (BD2)-selective BET inhibitor with pIC50 7.9 (BRD4 BD2), 1260-fold selectivity over BRD4 BD1.
    GSK852 demonstrates highly soluble with good in vivo rat and dog pharmacokinetics.

    物理化学性质&存储条件

    分子量 406.482
    分子式 C24H26N2O4
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (3S)-N5-((1R,3R,5S)-3-hydroxybicyclo[3.1.0]hexan-6-yl)-N7,3-dimethyl-3-phenyl-2,3-dihydrobenzofuran-5,7-dicarboxamide

    参考文献

    1. Simon C C Lucas, et al. J Med Chem. 2021 Aug 12;64(15):10711-10741.

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