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首页-小分子抑制剂&激动剂-Epigenetics-Bromodomain-GSK789
GSK789

Chemical Structure : GSK789

CAS No.: 2540591-06-6

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GSK789 (GSK-789)

货号: PC-72470Not For Human Use, Lab Use Only.

GSK789 (GSK-789) is a potent, cell-permeable, and highly selective inhibitor of the first bromodomains (BD1) of the BET family with IC50 of 20 nM BRD4 BD1, 1500-fold selectivity over BD2.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    GSK789 (GSK-789) is a potent, cell-permeable, and highly selective inhibitor of the first bromodomains (BD1) of the BET family with IC50 of 20 nM BRD4 BD1, 1500-fold selectivity over BD2.

    物理化学性质&存储条件

    分子量 463.582
    分子式 C26H33N5O3
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (3R,4R)-N-cyclohexyl-4-((5-(furan-2-yl)-3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)-1-methylpiperidine-3-carboxamide

    参考文献

    1. Robert J Watson, et al. J Med Chem. 2020 Sep 10;63(17):9045-9069.

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