GSK3011724A | KasA inhibitor | Probechem Biochemicals

Chemical Structure : GSK3011724A

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GSK3011724A (DG167;GSK-3011724;GSK-724A;GSK-724)

货号: PC-35948Not For Human Use, Lab Use Only.

GSK3011724A (DG167, GSK3011724A) is a potent, specific inhibitor of β-ketoacyl-ACP synthase (KasA, Kd=9 nM), shows anti-tubercular activity (MIC H37Rv=0.8 uM).

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生物&药学活性

GSK3011724A (DG167, GSK3011724A) is a potent, specific inhibitor of β-ketoacyl-ACP synthase (KasA, Kd=9 nM), shows anti-tubercular activity (MIC H37Rv=0.8 uM).
GSK3011724A (DG167) shows much weaker apparent dissociation constant for both Pks10 and Pks (Kd=1.4 uM).
GSK3011724A (DG167) inhibits mycolic acid biosynthesis and shows negligible activity against a panel of unrelated proteins and 18 Gram-positive and Gram-negative bacterial species.

物理化学性质&存储条件

分子量	267.347
分子式	C12H17N3O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(1-methyl-1H-indazol-6-yl)butane-1-sulfonamide

参考文献

1. Kumar P, et al. MBio. 2018 Dec 18;9(6). pii: e02101-17.

2. Abrahams KA, et al. Nat Commun. 2016 Sep 1;7:12581.

GSK3011724A (DG167;GSK-3011724;GSK-724A;GSK-724)

生物&药学活性

物理化学性质&存储条件

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GSK3011724A (DG167;GSK-3011724;GSK-724A;GSK-724)

生物&药学活性

物理化学性质&存储条件

参考文献

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