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首页-小分子抑制剂&激动剂-Others-GRK (GPCRK)-GSK180736A
GSK180736A

Chemical Structure : GSK180736A

CAS No.: 817194-38-0

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GSK180736A (GSK 180736A, GSK-180736A)

货号: PC-45590Not For Human Use, Lab Use Only.

GSK180736A is a highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM.

规格 价格 库存 数量
5 mg (Free Sample) ￥280 In stock
10 mg ￥780 In stock
25 mg ￥1380 In stock
50 mg ￥2480 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GSK180736A is a highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM.
GSK180736A displays >400-fold selective for GRK2 over both GRK1 and GRK5, with no inhibition on PKA; also inhibits ROCK with IC50 of 0.1 uM.

物理化学性质&存储条件

分子量 365.3611
分子式 C19H16FN5O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: ≥ 30 mg/mL
Chemical Name/SMILES

5-Pyrimidinecarboxamide, 4-(4-fluorophenyl)-1,2,3,4-tetrahydro-N-1H-indazol-5-yl-6-methyl-2-oxo-

参考文献

1. Homan KT, et al. ACS Chem Biol. 2015 Jan 16;10(1):310-9.

2. Waldschmidt HV, et al. J Med Chem. 2016 Apr 28;59(8):3793-807.

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