GSK1379725A |CAS:1802251-00-8 Probechem Biochemicals

Chemical Structure : GSK1379725A

CAS No.: 1802251-00-8

加入收藏

GSK1379725A (GSK 1379725A, BPTF inhibitor AU1)

货号: PC-62389Not For Human Use, Lab Use Only.

GSK1379725A is the first selective small molecule inhibitor of BPTF bromodomain (bromodomain PHD finger transcription factor) with Kd of 2.8 uM in a cell-based reporter assay, shows no binding activity for Brd4.

规格	价格	库存
5 mg	￥1980	In stock
10 mg	￥3180	In stock
25 mg	￥5280	In stock
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

GSK1379725A is the first selective small molecule inhibitor of BPTF bromodomain (bromodomain PHD finger transcription factor) with Kd of 2.8 uM in a cell-based reporter assay, shows no binding activity for Brd4.
GSK1379725A interferes with its regulatory activity in cultured cells.

物理化学性质&存储条件

分子量	450.47
分子式	C23H23FN6O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzoic acid, 3-[[[[1-[2-[(4-fluorophenyl)amino]-4-pyrimidinyl]-3-pyrrolidinyl]amino]carbonyl]amino]-, methyl ester

参考文献

1. Urick AK, et al. ACS Chem Biol. 2015 Oct 16;10(10):2246-56.

GSK1379725A (GSK 1379725A, BPTF inhibitor AU1)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

GSK1379725A (GSK 1379725A, BPTF inhibitor AU1)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.