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首页-小分子抑制剂&激动剂-Epigenetics-Bromodomain-GSK1379725A
GSK1379725A

Chemical Structure : GSK1379725A

CAS No.: 1802251-00-8

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GSK1379725A (GSK 1379725A, BPTF inhibitor AU1)

货号: PC-62389Not For Human Use, Lab Use Only.

GSK1379725A is the first selective small molecule inhibitor of BPTF bromodomain (bromodomain PHD finger transcription factor) with Kd of 2.8 uM in a cell-based reporter assay, shows no binding activity for Brd4.

规格 价格 库存 数量
5 mg ￥1280 In stock
10 mg ￥1980 In stock
25 mg ￥3580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GSK1379725A is the first selective small molecule inhibitor of BPTF bromodomain (bromodomain PHD finger transcription factor) with Kd of 2.8 uM in a cell-based reporter assay, shows no binding activity for Brd4.
GSK1379725A interferes with its regulatory activity in cultured cells.

物理化学性质&存储条件

分子量 450.47
分子式 C23H23FN6O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Benzoic acid, 3-[[[[1-[2-[(4-fluorophenyl)amino]-4-pyrimidinyl]-3-pyrrolidinyl]amino]carbonyl]amino]-, methyl ester

参考文献

1. Urick AK, et al. ACS Chem Biol. 2015 Oct 16;10(10):2246-56.

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