GSK-5959 |CAS:901245-65-6 Probechem Biochemicals

Chemical Structure : GSK-5959

CAS No.: 901245-65-6

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GSK-5959 (GSK5959, GSK 5959)

货号: PC-45508Not For Human Use, Lab Use Only.

GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.

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10 mg	￥1280	In stock
25 mg	￥2180	In stock
50 mg	￥3780	In stock
100 mg		Get quote

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GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.
GSK-5959 shows about 2 logs selectivity over BRPF2/3 and less potent for BRD4 (pIC50<4.3).

物理化学性质&存储条件

分子量	394.4668
分子式	C22H26N4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: < 7.8 mg/mL
Chemical Name/SMILES	Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-

参考文献

1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.

GSK-5959 (GSK5959, GSK 5959)

生物&药学活性

物理化学性质&存储条件

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GSK-5959 (GSK5959, GSK 5959)

生物&药学活性

物理化学性质&存储条件

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