GSK-114 |CAS:1301761-96-5 Probechem Biochemicals

Chemical Structure : GSK-114

CAS No.: 1301761-96-5

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GSK-114 (GSK114)

货号: PC-62726Not For Human Use, Lab Use Only.

GSK-114 is a potent, selective TNNI3K (TNNI3 Interacting Kinase) inhibitor with IC50 of 25 nM, dispalys 40-fold over B-Raf, exceptional broad spectrum kinase selectivity (IC50>1,000 nM, 99% of kinases, 291/294).

规格	价格	库存
5 mg	￥1380	In stock
10 mg	￥2180	In stock
25 mg	￥3480	In stock
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

GSK-114 is a potent, selective TNNI3K (TNNI3 Interacting Kinase) inhibitor with IC50 of 25 nM, dispalys 40-fold over B-Raf, exceptional broad spectrum kinase selectivity (IC50>1,000 nM, 99% of kinases, 291/294).
GSK-114 has adequate oral exposure to enable its use in cellular and in vivo studies.

物理化学性质&存储条件

分子量	417.484
分子式	C19H23N5O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-((6,7-dimethoxyquinazolin-4-yl)amino)-4-(dimethylamino)-N-methylbenzenesulfonamide

参考文献

1. Lawhorn BG, et al. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3355-8.

GSK-114 (GSK114)

生物&药学活性

物理化学性质&存储条件

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GSK-114 (GSK114)

生物&药学活性

物理化学性质&存储条件

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