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首页-小分子抑制剂&激动剂-GPCR-Neurokinin Receptor-GR-64349
GR-64349

Chemical Structure : GR-64349

CAS No.: 137593-52-3

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GR-64349 (GR64349)

货号: PC-63098Not For Human Use, Lab Use Only.

GR-64349 is a potent and selective tachykinin NK2 receptor (NK2R) agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GR-64349 is a potent and selective tachykinin NK2 receptor (NK2R) agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.

物理化学性质&存储条件

分子量 921.12
分子式 C42H68N10O11S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

KDSFVGLM (Modifications: Leu-7 = R-γ-lactam-Leu, Met-8 = C-terminal amide)

参考文献

1. Deal MJ, et al. J Med Chem. 1992 Oct 30;35(22):4195-204.

2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.

3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.

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