GPR7 antagonist 21a

Chemical Structure : GPR7 antagonist 21a

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货号: PC-38613Not For Human Use, Lab Use Only.

GPR7 antagonist 21a is a highly potent small molecule antagonist of NPBWR1 (GPR7) antagonist with cAMP IC50 of 30 nM, dose-dependently increased [125I]-hNPW23 dissociation rate constants from NPBWR1 in kinetic binding assays.

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生物&药学活性

GPR7 antagonist 21a is a highly potent small molecule antagonist of NPBWR1 (GPR7) antagonist with cAMP IC50 of 30 nM, dose-dependently increased [125I]-hNPW23 dissociation rate constants from NPBWR1 in kinetic binding assays.

物理化学性质&存储条件

分子量	397.182
分子式	C17H9Cl2F3N4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(2,6-dichloro-4-(1H-pyrazol-4-yl)phenyl)-5-(trifluoromethyl)-1H-benzo[d]imidazole

参考文献

1. Remond Moningka, et al. Bioorg Med Chem Lett. 2020 Dec 1;30(23):127510.