GPR61 inverse agonist 15

Chemical Structure : GPR61 inverse agonist 15

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货号: PC-26403Not For Human Use, Lab Use Only.

GPR61 inverse agonist 15 is a potent, selective, and brain-penetrant GPR61 inverse agonist with cAMP functional IC50 of 6.2 nM and 20 nM for human and mouse GPR61 respectively.

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生物&药学活性

GPR61 inverse agonist 15 is a potent, selective, and brain-penetrant GPR61 inverse agonist with cAMP functional IC50 of 6.2 nM and 20 nM for human and mouse GPR61 respectively.

物理化学性质&存储条件

分子量	454.88
分子式	C18H17ClF2N6O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(5-Chloro-4,6-dimethylpyrimidin-2-yl)-6-(((3,5-difluoropyridin-4-yl)methyl)amino)-2-methylpyridine-3-sulfonamide

参考文献

1. Fisher EL, et al. J Med Chem. 2026 Mar 15. doi: 10.1021/acs.jmedchem.6c00081.