GPR55 agonist 28

Chemical Structure : GPR55 agonist 28

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货号: PC-21153Not For Human Use, Lab Use Only.

GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays.

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生物&药学活性

GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays.
GPR55 agonist 28 activates the β-arrestin pathway with EC50 of 6.2 nM, produces a full activation of hGPR55 in the Ca2+ flux assay (Emax: 105%).
GPR55 agonist 28 (10 uM) markedly decreased the frequency of rat MSN cell firing in cultured rodent striatal MSNs.

物理化学性质&存储条件

分子量	365.37
分子式	C19H16FN5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-5-(3-((1-(4-Fluorophenyl)ethyl)amino)-1,2,4-triazin-6-yl)-3-methylbenzo[d]oxazol-2(3H)-one

参考文献

1. Richard C. Hewer, et al. J. Med. Chem. 2023.

GPR55 agonist 28

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物理化学性质&存储条件

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GPR55 agonist 28

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物理化学性质&存储条件

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