GPR39 agonist 7 |CAS:1582736-32-0 Probechem Biochemicals

Chemical Structure : GPR39 agonist 7

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GPR39 agonist 7

货号: PC-62256Not For Human Use, Lab Use Only.

GPR39 agonist 7 is a Hedgehog pathway inhibitor that has high cellular potency (EC50=20 nM) in the reporter gene assay, activates the orphan receptor GPR39 and potently reduces of Gli1 and Ptch1 mRNA levels.

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GPR39 agonist 7 is a Hedgehog pathway inhibitor that has high cellular potency (EC50=20 nM) in the reporter gene assay, activates the orphan receptor GPR39 and potently reduces of Gli1 and Ptch1 mRNA levels.
GPR39 agonist 7 activates the orphan receptor GPR39, which signals to the Gli transcription factors and blocks signaling.
GPR39 agonist 7 is a useful chemical tool for in vitro interrogation of GPR39 signaling in different cellular contexts.

物理化学性质&存储条件

分子量	604.774
分子式	C31H40N8O3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(5-((2-((((1r,4r)-4-(((3-cyanophenyl)sulfonamido)methyl)cyclohexyl)methyl)amino)-6-(pyridin-2-yl)pyrimidin-4-yl)amino)pentyl)acetamide

参考文献

1. Bassilana F, et al. Nat Chem Biol. 2014 May;10(5):343-9.

GPR39 agonist 7

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物理化学性质&存储条件

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GPR39 agonist 7

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物理化学性质&存储条件

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