GPR183 inverse agonist compound 78 | GPR183 inverse agonist

Chemical Structure : GPR183 inverse agonist compound 78

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GPR183 inverse agonist compound 78 (GPR183 inverse agonist 1)

货号: PC-27089Not For Human Use, Lab Use Only.

GPR183 inverse agonist 1 (Compound 78) is a seletive GPR183 (EBI-2) inverse agonist, inhibits the GPR183-mediated Gi activation with pIC50 of 6.29, modulates both Gi and β-arrestin2-responses of GPR183.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

GPR183 inverse agonist 1 (Compound 78) is a seletive GPR183 (EBI-2) inverse agonist, inhibits the GPR183-mediated Gi activation with pIC50 of 6.29, modulates both Gi and β-arrestin2-responses of GPR183.

物理化学性质&存储条件

分子量	442.32
分子式	C20H20BrN5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((1-(4-bromobenzoyl)piperidin-4-yl)methyl)-6-(1H-pyrazol-1-yl)pyridazin-3(2H)-one

参考文献

1. Andersson L, et al. Nat Commun. 2026 May 30. doi: 10.1038/s41467-026-73857-9.