GKM-001 | Glucokinase activator | Probechem Biochemicals

Chemical Structure : GKM-001

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GKM-001 (GKM001)

货号: PC-49837Not For Human Use, Lab Use Only.

GKM-001 is a potent, liver-selective small molecule activator of glucokinase (GKA), demonstrates glucose lowering effect without hypoglycemia in normal and type II diabetes mellitus (T2DM).

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

GKM-001 is a potent, liver-selective small molecule activator of glucokinase (GKA) with EC50 of 1.55 and 4.3 uM for human and rat GK, respectively.
GKM-001 demonstrates glucose lowering effect without hypoglycemia in normal and type II diabetes mellitus (T2DM).

物理化学性质&存储条件

分子量	580.02
分子式	C25H20ClF2N3O5S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(5-chloro-2-(1-(3,4-difluorobenzyl)-4-(4-(methylsulfonyl)benzyl)-1H-pyrrole-2-carboxamido)thiazol-4-yl)acetic acid

参考文献

1. Patent WO2008149382 A1.

GKM-001 (GKM001)

生物&药学活性

物理化学性质&存储条件

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GKM-001 (GKM001)

生物&药学活性

物理化学性质&存储条件

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