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首页-小分子抑制剂&激动剂-GPCR-Protease-activated Receptor (PAR)-GB-110
GB-110

Chemical Structure : GB-110

CAS No.: 1252806-70-4

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GB-110 (GB 110;GB110)

货号: PC-60319Not For Human Use, Lab Use Only.

GB-110 is a potent, non-peptidic agonist of PAR2 that selectively induces PAR2-mediated intracellular Ca(2+) release in HT29 cells with EC50 of 0.28 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

GB-110 is a potent, non-peptidic agonist of PAR2 that selectively induces PAR2-mediated intracellular Ca(2+) release in HT29 cells with EC50 of 0.28 uM.
GB-110 displays no activity for PAR-1 receptors.

物理化学性质&存储条件

分子量 608.784
分子式 C33H48N6O5
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-((S)-1-(((2S,3S)-1-((3-(4-(aminomethyl)piperidine-1-carbonyl)benzyl)amino)-3-methyl-1-oxopentan-2-yl)amino)-3-cyclohexyl-1-oxopropan-2-yl)isoxazole-5-carboxamide

参考文献

1. Barry GD, et al. J Med Chem. 2010 Oct 28;53(20):7428-40.

2. Suen JY, et al. Br J Pharmacol. 2012 Mar;165(5):1413-23.

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