GAT100 |CAS:1663564-42-8 Probechem Biochemicals

Chemical Structure : GAT100

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GAT100 (GAT-100)

货号: PC-35488Not For Human Use, Lab Use Only.

GAT-100 (GAT100) is a potent, selective CB1R negative allosteric modulator (NAM) with cAMP EC50 and β-arr EC50 of 174 nM and 2.1 nM, does not exhibit inverse agonism.

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生物&药学活性

GAT-100 (GAT100) is a potent, selective CB1R negative allosteric modulator (NAM) with cAMP EC50 and β-arr EC50 of 174 nM and 2.1 nM, does not exhibit inverse agonism.
GAT-100 is a covalent probe for mapping structure-function correlates characteristic of the druggable CB1R allosteric space.

物理化学性质&存储条件

分子量	432.59
分子式	C25H28N4OS
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-Ethyl-5-isothiocyanato-N-(4-(piperidin-1-yl)phenethyl)-1H-indole-2-carboxamide

参考文献

1. Kulkarni PM, et al. J Med Chem. 2016 Jan 14;59(1):44-60.

2. Laprairie RB, et al. ACS Chem Neurosci. 2016 Jun 15;7(6):776-98.

GAT100 (GAT-100)

生物&药学活性

物理化学性质&存储条件

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GAT100 (GAT-100)

生物&药学活性

物理化学性质&存储条件

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