GAP-134 | Gap-junction modifier | Probechem Biochemicals

Chemical Structure : GAP-134

CAS No.: 943134-39-2

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GAP-134 (Danegaptide, ZP1609, GAP134)

货号: PC-42735Not For Human Use, Lab Use Only.

GAP-134 (Danegaptide) is a potent, orally active gap-junction modifier, prevents significantly conduction velocity slowing at 10 nM compared with vehicle.

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10 mg	￥2480	In stock
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生物&药学活性

GAP-134 (Danegaptide) is a potent, orally active gap-junction modifier, prevents significantly conduction velocity slowing at 10 nM compared with vehicle.
GAP-134 (Danegaptide) has highly desirable in vitro and in vivo safety profile including (1) lack of direct effects on membrane ion currents, hERG inhibition, and CYP450 liabilities, (2) negative AMES result, (3) a benign NovaScreen profile, and (4) no effects on systemic hemodynamics.

物理化学性质&存储条件

分子量	291.3025
分子式	C14H17N3O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	L-Proline, glycyl-4-(benzoylamino)-, (4R)-

参考文献

1. Butera JA, et al. J Med Chem. 2009 Feb 26;52(4):908-11.

2. Rossman EI, et al. J Pharmacol Exp Ther. 2009 Jun;329(3):1127-33.

3. Hennan JK, et al. J Cardiovasc Pharmacol Ther. 2009 Sep;14(3):207-14.

GAP-134 (Danegaptide, ZP1609, GAP134)

生物&药学活性

物理化学性质&存储条件

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GAP-134 (Danegaptide, ZP1609, GAP134)

生物&药学活性

物理化学性质&存储条件

参考文献

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