GAK inhibitor 49 |CAS:319492-82-5 Probechem Biochemicals

Chemical Structure : GAK inhibitor 49

CAS No.: 319492-82-5

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GAK inhibitor 49

货号: PC-35412Not For Human Use, Lab Use Only.

GAK inhibitor 49 is a potent, selective, ATP-competitive inhibitor of cyclin G-associated kinase (GAK, cell IC50=56 nM) with favourable NAK family selectivity (AAK1, STK16, BMP2K).

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5 mg	￥1580	In stock
10 mg	￥2380	In stock
25 mg	￥3980	In stock
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生物&药学活性

GAK inhibitor 49 is a potent, selective, ATP-competitive inhibitor of cyclin G-associated kinase (GAK, cell IC50=56 nM) with favourable NAK family selectivity (AAK1, STK16, BMP2K).
GAK inhibitor 49 shows binding to only GAK and RIPK2 in an unbiased MIB/MS experiment in cell lysate.

物理化学性质&存储条件

分子量	370.405
分子式	C20H22N2O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine

参考文献

1. Asquith CRM, et al. ChemMedChem. 2018 Jan 8;13(1):48-66.

2. Pu SY, et al. J Med Chem. 2018 Jul 16. doi: 10.1021/acs.jmedchem.8b00613.

GAK inhibitor 49

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GAK inhibitor 49

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