G-9791 |CAS:1926204-95-6 Probechem Biochemicals

首页-小分子抑制剂&激动剂-Cell Cycle/DNA Damage-p21-activated Kinase (PAK)-G-9791

Chemical Structure : G-9791

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G-9791 (G 9791;G9791)

货号: PC-60221Not For Human Use, Lab Use Only.

G-9791 (G9791) is a potent and selective group I PAK (pan-PAK1/2/3) inhibitor with Ki of 0.95/2 nM for PAK1/2, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

G-9791 (G9791) is a potent and selective group I PAK (pan-PAK1/2/3) inhibitor with Ki of 0.95/2 nM for PAK1/2, respectively.
G-9791 displays 57-fold selectivity over Lck kinase.
G-9791 inhibits the phosphorylation of residue S298 of MEK1 in EBC1 cells with IC50 of 33 nM.

物理化学性质&存储条件

分子量	508.98
分子式	C26H26ClFN6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6-(2-Chloro-4-(3-methyl-2-oxopyridin-1(2H)-yl)phenyl)-8-(2-(3-fluoro-1-methylazetidin-3-yl)ethyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8H)-one

参考文献

1. Rudolph J, et al. J Med Chem. 2016 Jun 9;59(11):5520-41.

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G-9791 (G 9791;G9791)

生物&药学活性

物理化学性质&存储条件

参考文献

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G-9791 (G 9791;G9791)

生物&药学活性

物理化学性质&存储条件

参考文献

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