Feniralstat (KVD-824) | Kallikrein inhibitor | Probechem Biochemicals

Chemical Structure : Feniralstat

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Feniralstat (KVD-824, KVD824)

货号: PC-73418Not For Human Use, Lab Use Only.

Feniralstat (KVD-824) is a potent, selective kallikrein inhibitor with IC50 of 6.7 nM for human plasma kallikrein (pKal), dispays no inhibition against human KLKl, FXIa and Factor Xlla (IC50>40 uM).

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生物&药学活性

Feniralstat (KVD-824) is a potent, selective kallikrein inhibitor with IC50 of 6.7 nM for human plasma kallikrein (pKal), dispays no inhibition against human KLKl, FXIa and Factor Xlla (IC50>40 uM).

物理化学性质&存储条件

分子量	509.514
分子式	C26H25F2N5O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(4-((5-fluoro-2-oxopyridin-1(2H)-yl)methyl)benzyl)-N-((3-fluoro-4-methoxypyridin-2-yl)methyl)-3-(methoxymethyl)-1H-pyrazole-4-carboxamide

参考文献

1. Rebecca Louise DAVIE, et al. Pyrazole derivatives as plasma kallikrein inhibitors. WO2017207983A1. (Compound 30).

Feniralstat (KVD-824, KVD824)

生物&药学活性

物理化学性质&存储条件

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Feniralstat (KVD-824, KVD824)

生物&药学活性

物理化学性质&存储条件

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