Fasitibant | B2R antagonist | Probechem Biochemicals

Chemical Structure : Fasitibant

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Fasitibant (MEN16132, MEN-16132)

货号: PC-26631Not For Human Use, Lab Use Only.

Fasitibant (MEN16132) is a potent, selective, nonpeptide antagonist of type 2 bradykinin receptor (B2R) with pIC50 of 10.5 for [3H]-BK binding in mouse lung.

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生物&药学活性

Fasitibant (MEN16132) is a potent, selective, nonpeptide antagonist of type 2 bradykinin receptor (B2R) with pIC50 of 10.5 for [3H]-BK binding in mouse lung.

物理化学性质&存储条件

分子量	836.69
分子式	C36H50Cl4N6O6S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-4-amino-5-(4-(4-((2,4-dichloro-3-(((2,4-dimethylquinolin-8-yl)oxy)methyl)phenyl)sulfonamido)tetrahydro-2H-pyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-5-oxopentan-1-aminium chloride hydrochloride

参考文献

1. Valenti C, et al. Br J Pharmacol. 2012 Jun;166(4):1403-10.

2. Cialdai C, et al. J Pharmacol Exp Ther. 2009 Dec;331(3):1025-32.

3. Meini S, et al. Br J Pharmacol. 2007 Feb;150(3):313-20.

Fasitibant (MEN16132, MEN-16132)

生物&药学活性

物理化学性质&存储条件

参考文献

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Fasitibant (MEN16132, MEN-16132)

生物&药学活性

物理化学性质&存储条件

参考文献

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