FG-7142 (FG 7142, ZK 39106, LSU-65) | Benzodiazepine inverse agonist

Chemical Structure : FG-7142

CAS No.: 78538-74-6

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FG-7142 (ZK 39106, LSU-65, FG 7142, FG7142)

货号: PC-28085Not For Human Use, Lab Use Only.

FG-7142 (FG 7142, ZK 39106, LSU-65) is an anxiogenic benzodiazepine inverse agonist / antagonist, has high affinity for α1 subunit-containing GABAA receptor with Ki of 91 nM, also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit with EC50 of 137 nM.

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10 mg	￥580	In stock
25 mg	￥980	In stock
50 mg	￥1580	In stock
100 mg	￥2580	In stock
250 mg		Get quote

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FG-7142 (FG 7142, ZK 39106, LSU-65) is an anxiogenic benzodiazepine inverse agonist / antagonist, has high affinity for α1 subunit-containing GABAA receptor with Ki of 91 nM, also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit with EC50 of 137 nM.

物理化学性质&存储条件

分子量	225.25
分子式	C13H11N3O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-Methyl-9H-pyrido[3,4-b]indole-3-carboxamide

参考文献

1. Petersen EN, et al. Eur J Pharmacol. 1982 Aug 27;82(3-4):217-21.

2. Rossier J, et al. Lancet. 1983 Jan 1;1(8314-5):77-8.

3. Ongini E, et al. Eur J Pharmacol. 1983 Nov 11;95(1-2):125-9.

4. Cottone P, et al. Neuropsychopharmacology. 2007 May;32(5):1069-81.

FG-7142 (ZK 39106, LSU-65, FG 7142, FG7142)

生物&药学活性

物理化学性质&存储条件

参考文献

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FG-7142 (ZK 39106, LSU-65, FG 7142, FG7142)

生物&药学活性

物理化学性质&存储条件

参考文献

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