Euphol

Chemical Structure : Euphol

CAS No.: 514-47-6

加入收藏

货号: PC-25687Not For Human Use, Lab Use Only.

Euphol is a potent and reversible monoacylglycerol lipase (MAGL, MGL) inhibitor with IC50 of 315 nM (purified MGL).

规格	价格	库存
10 mg	￥680	In stock
25 mg	￥1080	In stock
50 mg	￥1780	In stock
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

Euphol is a potent and reversible monoacylglycerol lipase (MAGL, MGL) inhibitor with IC50 of 315 nM (purified MGL).
Euphol inhibits non-purified MGL (cell lysates of MGL-transfected HeLa cells) with IC50 of 882 nM.
Euphol inhibits MGL through a mechanism that is rapid, reversible and non-competitive, shows reversible interaction with Cys201 of MAGL.
Euphol protects 2-AG from degradation in intact rat brain neurons.

物理化学性质&存储条件

分子量	426.73
分子式	C30H50O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(3S,5R,10S,13S,14S,17S)-4,4,10,13,14-pentamethyl-17-((R)-6-methylhept-5-en-2-yl)-2,3,4,5,6,7,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-ol

参考文献

1. King AR, et al. Chem Biol. 2009 Oct 30;16(10):1045-52.

Euphol

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Euphol

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.