Eribaxaban |CAS:536748-46-6 Probechem Biochemicals

Chemical Structure : Eribaxaban

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Eribaxaban (PD-0348292;PD0348292;PD 0348292)

货号: PC-60954Not For Human Use, Lab Use Only.

A potent, selective and orally efficacious factor Xa (FXa) inhibitor with IC50 of 0.32 nM.

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生物&药学活性

A potent, selective and orally efficacious factor Xa (FXa) inhibitor with IC50 of 0.32 nM; displays >1,000-fold selectivity over a series of related serine proteases (thrombin, activated protein C, plasmin, tissue plasminogen activator and trypsin); potently inhibits thrombosis and shows potential for s for the treatment and prevention of thrombotic disorders.

Thrombosis

Phase 2 Discontinued

物理化学性质&存储条件

分子量	484.912
分子式	C24H22ClFN4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2R,4R)-1-N-(4-chlorophenyl)-2-N-[2-fluoro-4-(2-oxopyridin-1-yl)phenyl]-4-methoxypyrrolidine-1,2-dicarboxamide

参考文献

1. Kohrt JT, et al. Chem Biol Drug Des. 2007 Aug;70(2):100-12.

2. McBane RD 2nd, et al. Arterioscler Thromb Vasc Biol. 2008 Mar;28(3):413-8.

3. Karnicki K, et al. Thromb Haemost. 2008 Apr;99(4):759-66.

4. Cohen AT, et al. J Thromb Haemost. 2013 Aug;11(8):1503-10.

Eribaxaban (PD-0348292;PD0348292;PD 0348292)

生物&药学活性

物理化学性质&存储条件

参考文献

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Eribaxaban (PD-0348292;PD0348292;PD 0348292)

生物&药学活性

物理化学性质&存储条件

参考文献

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