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首页-小分子抑制剂&激动剂-Tyrosine Kinase-EGFR-Emupertinib
Emupertinib

Chemical Structure : Emupertinib

CAS No.: 2472802-77-8

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Emupertinib

货号: PC-24129Not For Human Use, Lab Use Only.

Emupertinib is a potent EGFR inhibitor with IC50 values of <0.3 nM, 0.52 nM, 0.5 nM, 0.69 nM and 0.92 nM for EGFR (d746-750/T790M/C779S), EGFR (L858R/T790M/C797S), EGFR (d746-750/C797S), EGFR (L858R/C797S), and EGFR (wild-type), respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

Emupertinib is a potent EGFR inhibitor with IC50 values of <0.3 nM, 0.52 nM, 0.5 nM, 0.69 nM and 0.92 nM for EGFR (d746-750/T790M/C779S), EGFR (L858R/T790M/C797S), EGFR (d746-750/C797S), EGFR (L858R/C797S), and EGFR (wild-type), respectively.

物理化学性质&存储条件

分子量 514.59
分子式 C30H26N8O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-(4-(4-amino-6-ethynyl-5-(quinolin-3-yl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[2.2.1]heptan-1-yl)-5-methylpyrazine-2-carboxamide

参考文献

1. Patent WO2023204304 A1.

2. Pantent WO2020166680 A1.

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