Eletriptan hydrobromide | 5-HT1B/1D agonist | Probechem Biochemicals

Chemical Structure : Eletriptan hydrobromide

CAS No.: 177834-92-3

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Eletriptan hydrobromide (UK 116044 hydrobromide, UK116044 hydrobromide)

货号: PC-61867Not For Human Use, Lab Use Only.

Eletriptan (UK 116044) hydrobromide is a potent, selective, and orally active 5-HT1B/1D receptor agonist with Ki of 0.92 nM and 3.14 nM respectively.

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25 mg	￥980	In stock
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100 mg	￥2480	In stock
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生物&药学活性

Eletriptan (UK 116044) hydrobromide is a potent, selective, and orally active 5-HT1B/1D receptor agonist with Ki of 0.92 nM and 3.14 nM respectively.
Eletriptan (UK 116044) significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease.
Eletriptan (UK 116044) displays antimigraine activity.

物理化学性质&存储条件

分子量	463.43
分子式	C22H26N2O2S.HBr
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide

参考文献

1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.

2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.

3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.

Eletriptan hydrobromide (UK 116044 hydrobromide, UK116044 hydrobromide)

生物&药学活性

物理化学性质&存储条件

参考文献

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Eletriptan hydrobromide (UK 116044 hydrobromide, UK116044 hydrobromide)

生物&药学活性

物理化学性质&存储条件

参考文献

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