Eletriptan (UK 116044) | 5-HT1B/1D agonist | Probechem Biochemicals

Chemical Structure : Eletriptan

加入收藏

Eletriptan (UK116044, UK 116044)

货号: PC-61868Not For Human Use, Lab Use Only.

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist with pKi of 8.0 and 8.9.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist with pKi of 8.0 and 8.9.
Eletriptan (UK 116044) significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease.
Eletriptan (UK 116044) displays antimigraine activity.

物理化学性质&存储条件

分子量	382.52
分子式	C22H26N2O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole

参考文献

1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.

2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.

3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.

Eletriptan (UK116044, UK 116044)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Eletriptan (UK116044, UK 116044)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.