Edoxaban tosylate monohydrate |CAS:1229194-11-9 Probechem Biochemicals

Chemical Structure : Edoxaban tosylate monohydrate

CAS No.: 1229194-11-9

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Edoxaban tosylate monohydrate

货号: PC-42504Not For Human Use, Lab Use Only.

A potent and orally active Factor Xa inhibitor with Ki of 0.561 nM.

规格	价格	库存
10 mg	￥1088.0	In stock
50 mg	￥4560	In stock
100 mg	￥7504.0	In stock

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生物&药学活性

A potent and orally active Factor Xa inhibitor with Ki of 0.561 nM; also inhibits prothrombinase (Ki=2.98 nM), weakly inhibits thrombin and FIXa (Ki=6.0 uM, and 41.7 uM); exhibits >10,000-fold selectivity for Fxa over FVIIa/sTF, FXIa, tPA, aPC, trypsin, plasmin and chymotrypsin; inhibits thrombus formation in rat and rabbit thrombosis models.

Thrombosis

Approved

物理化学性质&存储条件

分子量	738.2744
分子式	C31H40ClN7O8S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Ethanediamide, N1-(5-chloro-2-pyridinyl)-N2-[(1S,2R,4S)-4-[(dimethylamino)carbonyl]-2-[[(4,5,6,7-tetrahydro-5-methylthiazolo[5,4-c]pyridin-2-yl)carbonyl]amino]cyclohexyl]-, 4-methylbenzenesulfonate, hydrate (1:1:1)

参考文献

1. Furugohri T, et al. J Thromb Haemost. 2008 Sep;6(9):1542-9.

2. Furugohri T, et al. Eur J Pharmacol. 2012 Jul 5;686(1-3):74-80.

3. Morishima Y, et al. Thromb Res. 2013 Jan;131(1):59-63.

Edoxaban tosylate monohydrate

生物&药学活性

物理化学性质&存储条件

参考文献

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Edoxaban tosylate monohydrate

生物&药学活性

物理化学性质&存储条件

参考文献

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