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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Factor Xa-Edoxaban
Edoxaban

Chemical Structure : Edoxaban

CAS No.: 480449-70-5

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Edoxaban (DU-176)

货号: PC-42502Not For Human Use, Lab Use Only.

A potent and orally active Factor Xa inhibitor with Ki of 0.561 nM.

规格 价格 库存 数量
10 mg ￥2080 In stock
50 mg ￥7240 In stock
100 mg ￥9680 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

A potent and orally active Factor Xa inhibitor with Ki of 0.561 nM; also inhibits prothrombinase (Ki=2.98 nM), weakly inhibits thrombin and FIXa (Ki=6.0 uM, and 41.7 uM); exhibits >10,000-fold selectivity for Fxa over FVIIa/sTF, FXIa, tPA, aPC, trypsin, plasmin and chymotrypsin; inhibits thrombus formation in rat and rabbit thrombosis models.

Thrombosis

Approved

物理化学性质&存储条件

分子量 548.0575
分子式 C24H30ClN7O4S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Ethanediamide, N1-(5-chloro-2-pyridinyl)-N2-[(1S,2R,4S)-4-[(dimethylamino)carbonyl]-2-[[(4,5,6,7-tetrahydro-5-methylthiazolo[5,4-c]pyridin-2-yl)carbonyl]amino]cyclohexyl]-

参考文献

1. Furugohri T, et al. J Thromb Haemost. 2008 Sep;6(9):1542-9.

2. Furugohri T, et al. Eur J Pharmacol. 2012 Jul 5;686(1-3):74-80.

3. Morishima Y, et al. Thromb Res. 2013 Jan;131(1):59-63.

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