EZH2-IN-3 |CAS:1377997-28-8 Probechem Biochemicals

Chemical Structure : EZH2-IN-3

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EZH2-IN-3

货号: PC-62468Not For Human Use, Lab Use Only.

EZH2-IN-3 is a highly selective small molecule inhibitor of EZH2 and EZH1 with IC50 of 21/197/213 nM for wt EZH2/EZH2 Y641N/wt EZH1 respectively.

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生物&药学活性

EZH2-IN-3 is a highly selective small molecule inhibitor of EZH2 and EZH1 with IC50 of 21/197/213 nM for wt EZH2/EZH2 Y641N/wt EZH1 respectively.
EZH2-IN-3 suppresses global histone H3-lysine 27 methylation and cause selective proliferation defects.

物理化学性质&存储条件

分子量	490.004
分子式	C27H28ClN5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-chloro-4-(2-cyano-3-(pyridazin-4-yl)phenoxy)-N-(2,2,6,6-tetramethylpiperidin-4-yl)benzamide

参考文献

1. Garapaty-Rao S, et al. Chem Biol. 2013 Nov 21;20(11):1329-39.

EZH2-IN-3

生物&药学活性

物理化学性质&存储条件

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EZH2-IN-3

生物&药学活性

物理化学性质&存储条件

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