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首页-小分子抑制剂&激动剂-GPCR-Dopamine Receptor-ESG-1-60
ESG-1-60

Chemical Structure : ESG-1-60

CAS No.: 2899250-94-1

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ESG-1-60

货号: PC-24331Not For Human Use, Lab Use Only.

ESG-1-60 is a potent, selective partial agonist of dopamine D3 receptor (D3R) with Ki of 0.14 nM, EC50 of 3.43 nM (Go activation) and 0.2 nM (β-arrestin2 recruitment), show ~20-fold binding selectivity for D3 over D2 receptors.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

ESG-1-60 is a potent, selective partial agonist of dopamine D3 receptor (D3R) with Ki of 0.14 nM, EC50 of 3.43 nM (Go activation) and 0.2 nM (β-arrestin2 recruitment), show ~20-fold binding selectivity for D3 over D2 receptors.

物理化学性质&存储条件

分子量 442.43
分子式 C22H33Cl2N3O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Propanamide, N-[trans-4-[2-[4-(2,3-dichlorophenyl)-1-piperazinyl]ethyl]cyclohexyl]-3-methoxy-

参考文献

1. Soler-Cedeño O, et al. Br J Pharmacol. 2025 Mar 27. doi: 10.1111/bph.70021.

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