EPZ028862 | SMYD3 inhibitor | Probechem Biochemicals

Chemical Structure : EPZ028862

加入收藏

货号: PC-21039Not For Human Use, Lab Use Only.

EPZ028862 is a potent, selective inhibitor of SMYD3 with biochemical IC50 of 1.8 nM, and function of cellular methylation IC50 of 32 nM.

获取报价单

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

EPZ028862 is a potent, selective inhibitor of SMYD3 with biochemical IC50 of 1.8 nM, and function of cellular methylation IC50 of 32 nM.

分子量	422.54
分子式	C20H30N4O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C(C1=NOC(C2CC2)=C1)NC3CC(N4S(=O)([C@H]5CC[C@H](N)CC5)=O)CCC4C3

1. Michael J Thomenius, et al. PLoS One. 2018 Jun 1;13(6):e0197372.