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首页-小分子抑制剂&激动剂-GPCR-Mas-related G protein-coupled receptor (MRGPR)-EP-3945
EP-3945

Chemical Structure : EP-3945

CAS No.: 3057176-00-5

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EP-3945 (EP3945)

货号: PC-23536Not For Human Use, Lab Use Only.

EP-3945 is a potent, selective Mas-related G protein-coupled receptor MRGPRD agonist with EC50 of 211.6 nM at Gq in BRET assay, inactive against over 300 GPCRs.

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25 mg ￥7580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

EP-3945 is a potent, selective Mas-related G protein-coupled receptor MRGPRD agonist with EC50 of 211.6 nM at Gq in BRET assay, inactive against over 300 GPCRs.
EP-3945 activates MRGPRD much more potently than β-alanine and GABA.

物理化学性质&存储条件

分子量 418.50
分子式 C24H26N4O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-((1-(1-(4-methoxyphenyl)cyclopropane-1-carbonyl)piperidin-4-yl)amino)quinazolin-4(3H)-one

参考文献

1. Wang C, et al. Cell Rep. 2024 Nov 23;43(12):114942.

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