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首页-小分子抑制剂&激动剂-GPCR-Mas-related G protein-coupled receptor (MRGPR)-EP-2825
EP-2825

Chemical Structure : EP-2825

CAS No.: 958571-34-1

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EP-2825 (EP2825)

货号: PC-23537Not For Human Use, Lab Use Only.

EP-2825 is a potent, selective Mas-related G protein-coupled receptor MRGPRD agonist with EC50 of 211.6 nM at Gq in BRET assay.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

EP-2825 is a potent, selective Mas-related G protein-coupled receptor MRGPRD agonist with EC50 of 211.6 nM at Gq in BRET assay.
EP-2825 displays low off-target activity at SSTR4 and GPR97 in a panel of 300 GPCRs.
EP-2825 activates MRGPRD much more potently than β-alanine and GABA.

物理化学性质&存储条件

分子量 428.96
分子式 C23H29ClN4O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-((1-(2-(4-chlorophenyl)-2-methylpropanoyl)piperidin-4-yl)amino)-5,6,7,8-tetrahydroquinazolin-4(3H)-one

参考文献

1. Wang C, et al. Cell Rep. 2024 Nov 23;43(12):114942.

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