EHP-101 |CAS:1818428-24-8 Probechem Biochemicals

Chemical Structure : EHP-101

CAS No.: 1818428-24-8

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EHP-101 (Etrinabdione, VCE-004.8)

货号: PC-38051Not For Human Use, Lab Use Only.

EHP-101 (Etrinabdione, VCE-004.8) is an orally active, specific PPARγ and CB2 receptor dual agonist.

规格	价格	库存
5 mg	￥2280	In stock
10 mg	￥3580	In stock
25 mg	￥4980	In stock
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

EHP-101 (Etrinabdione, VCE-004.8) is an orally active, specific PPARγ and CB2 receptor dual agonist.
EHP-101 could prevent macrophage infiltration as well as the expression of Tenascin C (TNC), vascular cell adhesion molecule 1 (VCAM1), and the α-smooth muscle actin (SMA).
EHP-101 also prevent the reduced expression of vascular CD31 typical of skin fibrosis.
EHP-101 alleviates bleomycin-induced skin and lung fibrosis in mice.

物理化学性质&存储条件

分子量	433.592
分子式	C28H35NO3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1'R,6'R)-3-(benzylamino)-6-hydroxy-3'-methyl-4-pentyl-6'-(prop-1-en-2-yl)-[1,1'-bi(cyclohexane)]-2',3,6-triene-2,5-dione

参考文献

1. García-Martín A, et al. Biochem Pharmacol. 2018 Nov;157:304-313.

2. Navarrete C, et al. Neurobiol Dis. 2020 Sep;143:104994.

3. García-Martín A, et al. Biomed Pharmacother. 2021 Oct;142:112007.

EHP-101 (Etrinabdione, VCE-004.8)

生物&药学活性

物理化学性质&存储条件

参考文献

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EHP-101 (Etrinabdione, VCE-004.8)

生物&药学活性

物理化学性质&存储条件

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